chemical-categories

 

Pharmaceutical Grade Treatment Of Prostate Cancer Peptide Deslorelin Acetate 57773-65-6

 

Deslorelin Basic Info.:

 

Product Name: Deslorelin

Specification: 50mg*50vials/kit

Synonyms: GLP-HIS-TRP-SER-TYR-D-TRP-LEU-ARG-PRO-NHET;Desorelin;Deslorelin; Deslorelin Acetate; Deslorelin (Human);

CAS: 57773-65-6

MF: C64H83N17O12

MW: 1282.45

Purity: 98%

Storage temp.: −20°C

Product Categories: Peptide;Hormones

Usage: Biochemical research;Clinical used in the treatment of prostate cancer.

 

Deslorelin Description:

 

Deslorelin acetate is an injectable gonadotropin releasing hormone super-agonist (GnRH agonist) also known as an LHRH agonist. It stops the production of sex hormones (and oestrogen). Deslorelin Acetate is marketed by Peptech with the brand name Ovuplant. It is currently approved for use in veterinary medicine and is used to induce ovulation in mares as part of the artificial insemination process. It is also used to stabilize high-risk pregnancies, mainly of livestock. Unlike other GnRH agonists, which are mainly used to inhibit uteinizing hormone and follicle-stimulating hormone by their ultimate downregulation of the pituitary gland, Deslorelin is primarily used for the initial flare effect upon the pituitary, and its associated surge of LH secretion.

 

Deslorelin Application:

 

Deslorelin was successfully trialed in the US and was approved for veterinary use under certain  circumstances. In Europe, it was approved for use in equine assisted reproduction. It is also being trialed in humans to study its efficacy in treatment of breast cancer in women,and in treating  precocious puberty and congenital adrenal hyperplasia in male and female children.

 

 

Pharmaceutical Raw Materials Natural Steroid Hormones Powder Methyldienedione 5173-46-6

 

Methyldienedione Basic Info.:

 

Product Name: Methyldienedione

Alias: Estra-4,9-diene-3,17-dione

CAS register number: 5173-46-6

Molecular Formula: C18H22O2

Molecular Weight: 270.37

Melting Point: 131-134°C

Assay: 98%min

Grade: Pharmaceutical Grade

Storage: Shading, confined preservation

Packing: 1kg/foil bag. 25kg/drum

Character: White crystalline powder.

Usage: A potential metabolitie of STS 557 (Dienogest). A steroid with antiglucocorticoid activity.

 

Methyldienedione Description:

 

Estra-4,9-diene-3,17-dione is a powerful pro-steroid chemically similar to the anabolic agent Trenbolone.

When in the body, estra-4,9-diene-3,17-dione completes the conversion to Trenbolone. Trenbolone is a potent anabolic steroid, which binds to specific receptors present in reproductive tissue, muscle and fat.

 

Estra Diene Dione (estra-4,9-diene-3,17-dione) is an anabolic steroid and a precursor to Estra Diene Dione. It became a controlled substance in the US on January 4, 2010, and is classified as a Schedule III anabolic steroid under the United States Controlled Substances Act. Previous to this, it was sold as a bodybuilding supplement within the United States, and often mistakenly marketed as a prohormone for trenbolone, a veterinary steroid. Prior to its scheduling, it was part of a number of supplements that were seized during FDA enforcement for selling unapproved new drugs. The actual target steroid, Estra Diene Dione has some structural similarity to trenbolone, but lacks the 11-carbon -ene bond.

 

Methyldienedione Applications:

 

1. Protection from gynomastia,

2. Increased sex drive/libido,

3. Enhanced intensity & focus,

4. Estrogen control,

5. Positive effects on strength & lean mass.

 

 

Bodybuilding Supplements Anabolic Steroids Powder Mestanolone For Muscle Growth 521-11-9

 

Mestanolone Basic Info.:

 

Product Name: Mestanolone

Synonyms: Mestanolone;Mestaline;Methyldihydrotestosterone;Methylandrostanolone;17Alpha-Methyldihydrotestosterone;

CAS: 521-11-9

MF: C20H32O2

MW: 304.47

EINECS: 208-302-6

Melting point: 191°C

Storage temp.: Controlled Substance, -20°C Freezer

Appearance: White crystalline powder, Soluble in acetone, ethanol, ethyl acetate, insoluble in water.

Assay: 99%

Usage: Anabolic steroid. Controlled substance.

Product Categories: Steroids;Biochemistry;Hydroxyketosteroids;Intermediates & Fine Chemicals;Pharmaceuticals;Steroid and Hormone;API

 

Mestanolone Description: 

 

Mestanolone is the 17-methylated version of dihydrotestosterone (DHT). It is an orally bio-available androgenic steroid that is highly androgenic while only slightly anabolic. It is incapable of aromatization and it is not an agonist of the progesterone receptor.

Women should avoid Mestanolone for it is very androgenic. Long term use of it, say, more than 12 weeks should be avoided do to hepatoxicity. Since Mestanolone is unable to convert to estrogen, it is very useful during cutting phases or when one wishes to avoid excess weight gain.

Methyl DHT cannot convert to estrogen, but it does bind strongly to SHBG which can displace estrogen into circulation possibly resulting in estrogenic side effects.  

 

Mestanolone Applications:

 

Mestanolone is an anabolic steroid which are a group of drugs that are usually synthesized from the male reproduction hormone testosterone, and it can helps to rebuild body tissue, increase body and bone mass and encourage the formation of red blood cells.

It also is capable in increasing muscle strength and size, increasing muscle hardness, and also decrease body fat. They additionally reduce the fatigue associated with training, and the time required to recover after physical exertion. 

 

 

Healthy Weight Loss Drug Acomplia Steroids Powder Rimonabant For Fat Burning 168273-06-1

 

Rimonabant Basic info:

 

Product Name: Rimonabant

Synonyms: Acomplia; Rimonabant; SR141716; A 281; Sr 141716

CAS: 168273-06-1

Molecular formula: C22H21Cl3N4O

Molecular weight: 500.25

Purity: ≥ 99% by HPLC

Appearance: White crystalline powder

Package: 1kg/aluminium foil bag or as required

Professional team special for package and shipment and on tracking code 24hours for customs pass guaranteed.

 

Rimonabant Description:

 

An experimental wonder drug, Rimonabant, helps you lose weight, quit smoking and it also helps protect your heart. Trials have shown that 33% of people on Rimonabant lost 10% of body weight and kept their weight down for two years - this is a record, no other diet drug has managed to keep a person's weight down for so long. The second 33% lost 5% of body weight and kept it down. As well as keeping you lean, the drug also helps you quit the smoking habit. This will be of great interest for many smokers who are afraid to give up because they say they will put on loads of weight if they do

 

Rimonabant Brief Introduction:

 

Rimonabant has also been shown to be a μ-opioid receptor antagonist (possibly the contributing factor in its reported dysphoric qualities).Its main effect is reduction in appetite.

 

Rimonabant Application:

 

1. Obesity:

In a 2006 (2 year) study reported in JAMA, "Compared with the placebo group, the 20 mg of rimonabant group produced greater mean (SEM) reductions in weight (-6.3kg vs -1.6kg; P<.001), waist circumference (-6.1cm vs -2.5cm; P<.001), and level of triglycerides (percentage change, -5.3vs 7.9; P<.001) and a greater increase in level of high-density lipoprotein cholesterol (percentage change, 12.6vs 5.4; P<.001)."

 

2. Smoking cessation:

Rimonabant may also be found to be effective in assisting some smokers to quit smoking. Sanofi is currently conducting studies to determine the possible value of rimonabant in smoking-cessation therapy. The Studies with Rimonabant and Tobacco Use (STRATUS) program involves more than 6,000 subjects.

STRATUS is designed to explore two smoking-related therapies: first, to use rimonabant directly to aid in smoking cessation; second, to help prevent weight gain in former smokers. Initial results apparently suggest rimonabant is effective for both uses. However, the FDA has explicitly stated to Sanofi that, without additional studies, rimonabant cannot be approved in the United States for smoking cessation therapy.

 

 

Male Hormone Fitness Anabolic Steroids Powder Nandrolone Undecylate / Dynabolon 862-89-5

 

Nandrolone Undecylate Basic Info.:

 

Product Name: Nandrolone Undecylate

Synonyms: Nandrolone Undecanoate; Nandrolone 17β-Undecanoate;Dynabolon

CAS: 862-89-5

MF: C29H46O3

MW: 442.68

EIENCS: 212-729-3

Assay: 99% min.

Packing: foil bag or tin.

Delivery: Express courier.

Usage: pharmaceutical material, Tibolone intermediate.

Standard: Enterprise standard

 

Nandrolone Undecylate Description: 

 

Nandrolone undecylate is an effective compound that produces quality, long-lasting muscle gains. This is because of the relatively long half-life of the drug (around 8 days). Users report mild side effects, with the biggest side effect being water retention. 

 

Nandrolone Undecylate Applications:

 

Nandrolone is most commonly found with a cypionate, laurate, decanoate or plenylpropionate ester. Briefly explained, the ester determines how much of the given hormone is released over a period of time. Longer esters such as decanoate peak slowly and can keep stable blood plasma levels up to ten days, shorter esters such as the phenylpropionate peak more rapidly but the half-live is shorter. Shorter esters usually release much more active hormone per mg than longer esters, and of course, allow the drugs effects to leave your system more quickly.

 

 

Natural Herb Sex Enhancer Icariin / Horny Goat Weed Extract / Epimedium Extract 489-32-7

 

Epimedium Extract Basic Info:

 

Product Name: Epimedium Extract （Icariin）

Synonyms: Horny Goat Weed Extract;Icariin;Icarrin;Epimedium Extract;Epimedium Herb Ext;Epimedium P.E;Epimedium Brevicornum P.E;Epimedim Brevicormum P.E

CAS: 489-32-7

MF: C33H40O15

MW: 676.66

Melting point: 223-225 ºC

Density: 1.55

Storage temp.: room temp

Chemical Properties: Light yellow to yellow solid

Usage: hepatoprotective

Product Categories: Flavones;Functional Products;Natural Plant Extract;The group of Epimedii;plant extract;Nutritional Ingredients;Plant extracts;chemical reagent;pharmaceutical intermediate;phytochemical;reference standards from Chinese medicinal herbs (TCM).;standardized herbal extract;Standardized plant extract;Inhibitors;API

 

Epimedium Extract Description:

 

Epimedium as kidney tonifying herbs commonly used, can promote the effects of Epimedium on pituitary gonadal system function, can improve the male gonadal damage, increase the content of testosterone, but also promote the secretion of corticosterone and adrenal cortical cells. Reinforce the kidney yang effect of Herba Epimedii with its direct stimulation of target gland secretion of hormones involved. Epimedium can promote sexual function is due to hypersecretion of semen, seminal vesicle is filled, stimulation of sensory nerves, caused by indirect excited sexual desire.

 

Epimedium Extract Application:

 

Effect of Herba Epimedii from different aspects of aging mechanism, can delay the aging process and prevent the occurrence of senile disease. Such as the impact of cell passage, prolong the growth period, adjusting immunity and secretion system, improve metabolism and the function of various organs.

 

 

Oral or Injection Trenbolones Steroids 6-Bronmandrostenedione For Gain Muscle 38632-00-7

 

6-Bronmandrostenedione Basic Info.:

 

Product Name: 6-Bronmandrostenedione

Synonyms: (6b)-6-Bromoandrost-4-ene-3,17-dione; (6beta)-6-bromoandrost-4-ene-3,17-dione; 6-Bromoandrost-4-ene-3,17-dione

CAS RN.: 38632-00-7

Molecular Weight: 365.3046

Molecular Formula: C19H25BrO2

Density: 1.35g/cm3

Boiling Point(ºC): 467°C at 760 mmHg

Flash Point(ºC): 100.3°C

refractive_index: 1.577

Chemical Properties: Pale Yellow Solid

Usage: 6-Bronmandrostenedione analog, an aromatase inhibitor.

 

6-Bronmandrostenedione Description:

 

6-Bromodione is a fast acting competitive inhibitor of the aromatase enzyme. It works by binding to the aromatase enzyme to prevent it from aromatizing androgens. This is not a permanent binding and later acts to normalize aromatase (and thus estrogen levels) as hormone production returns to normal. It specifically targets aromatase and does not act as a central anti-androgen like some other post cycle products can. This means that your libido and mood will not be negatively affected.

 

6-Bronmandrostenedione Application:

 

6-beta-Bromodione works in a similar way but has an irreversible and permanent effect. This works well to mediate the excess aromatase that was produced while on cycle, while the alpha isomer works to normalize the natural levels. The goal is again to transition into normal production levels for all hormones affected by the anabolic cycle.

 

 

Pharmaceutical Raw Materials Female Steroids Raw Hormone Powders Mifepristone 84371-65-3

 

Mifepristone Basic Info.:

 

Product Name: Mifepristone (R38486)

Synonyms: 11-(4-(dimethylamino)phenyl)-17-hydroxy-17-(1-propynyl)-estra-9-dien-3-one;11beta-[4-(n,n-dimethylamino)phenyl]-17alpha-(prop-1-ynyl)-delta4,9-estradiene;r38486

CAS Number: 84371-65-3

Molecular Formula: C29H35NO2

Molecular Weight: 429.65

Assay: 99%

Melting Point: 195-198 °C

Storage temp.: 2-8°C

Appearance: Light yellowish powder

Product Categories: Steroids;Hormone;Acetylenes;Biochemistry;Functionalized Acetylenes;Hydroxyketosteroids;Chiral Reagents;Intermediates & Fine Chemicals;Pharmaceuticals;Intracellular receptor;Nuclear Receptors;Steroid and Hormone;API;Hormone Drugs.

Uses: It is a novel anti-progestin and has anti-glucocorticoid activity without the activity of progesterone, estrogen, androgen and anti-estrogen. It has a progesterone receptor affinity five times as high as progesterone. It is used for anti-pregnancy, inducing menstruation and terminating pregnancy, intrauterine inducer labor for dead fetal.

 

Mifepristone Description:

 

Mifepristone is a synthetic steroid compound with both antiprogesterone and antiglucocorticoid properties. The compound is a 19-nor steroid with substitutions at positions C11 and C17 (17 beta-hydroxy-11 beta-[4-dimethylamino phenyl] 17 alpha-[1-propynyl]estra-4, 9-dien-3-one), which antagonizes cortisol action competitively at the receptor level.

 

Mifepristone is a progesterone receptor antagonist used as an abortifacient in the first months of pregnancy, and in smaller doses as an emergency contraceptive. It is also a powerful glucocorticoid receptor antagonist.

 

Mifepristone Applications:

 

Mifepristone is used alone or in combination with misoprostol (Cytotec) to end an early pregnancy. Early pregnancy means it has been 49 days or less since your last menstrual period began. Mifepristone is in a class of medications called antiprogestational steroids. It works by blocking the activity of progesterone, a substance your body makes to help continue pregnancy.

 

Mifepristone is also available as another product (Korlym), which is used to control hyperglycemia (high blood sugar) in people with a certain type of Cushing's Syndrome in which the body makes too much of the hormone cortisol. This monograph only gives information about mifepristone (Mifeprex), which is used alone or in combination with another medication to end an early pregnancy. If you are using mifepristone to control hyperglycemia caused by Cushing's syndrome, read the monograph entitled mifepristone (Korlym) that has been written about this product.

 

Mifepristone (or RU-486) is a synthetic steroid compound with both antiprogesterone and antiglucocorticoid properties. The compound is a 19-nor steroid with substitutions at positions C11 and C17 (17 beta-hydroxy-11 beta-[4-dimethylamino phenyl] 17 alpha-[1-propynyl]estra-4, 9-dien-3-one), which antagonizes cortisol action competitively at the receptor level.

 

Mifepristone is a progesterone receptor antagonist used as an abortifacient in the first months of pregnancy, and in smaller doses as an emergency contraceptive. It is also a powerful glucocorticoid receptor antagonist, and has occasionally been used in refractory Cushing's syndrome (due to ectopic/neoplastic ACTH/cortisol secretion).

Mifepristone was the first antiprogestin to be developed and it has been evaluated extensively for its use as an abortifacient.

 

 

Safe Human Growth Hormone Peptide PT 141 Bremelanotide For Peptide Drum PT141 32780-32-8

 

PT 141 Basic Info.

 

Product Name: PT-141; PT141

CAS: 32780-32-8

MF: C50H69N15O10

MW: 1040.17736

Appearance: White powder

Water Content(Karl Fischer): ≤ 5.0%

Acetate Content(by HPLC): ≤ 15.0%

Amino Acid Composition: ± 10% of theoretical

Purity(by HPLC): ≥ 97.0%

Single Impurity(by HPLC): ≤ 1.0%

Peptide Content(by %N): ≥ 80%

Assay(By Anhydrous, Acetic Acid-free): 95.0~105.0%

Bacterial Endotoxins: ≤ 5EU/mg

Grade: Pharmceutical Grade

Storage: Shading, confined preservation

 

PT 141 Description:

 

PT-141 is a synthetic amino acid protein discovered during clinical trials using the Melanotan 2 for sunless tanning, photo-protection results from melanotans. Participants were documented as having experienced aphrodisiac reactions, leading to the further development PT-141. The melanocortin system targets receptors associated with desire through the melanocyte stimulating hormone paths that cross the blood-brain-barrier. Potentially the powerful sex-drug results feeling an aphrodisiac experience amplifying arousal pt141 reviews have shown the ability to increase libido effects of both men and women.

 

PT 141 Application:

 

PT-141 functions by activating the melanocortin receptor and MC4R namely. Bremelanotide originally was tested for nasal spray delivery but was discontinued after concerns about side effects. Bremelanotide PT141, as Melanotan II, may cause spontaneous arousal enhancing effect. Unlike other supplements, PT-141 results do not act on the vascular body, but directly increases desires through the nervous system.

 

 

Tesamorelin Anabolic Androgenic Steroids Tesamorelin Intramuscular Injection 218949-48-5

 

Tesamorelin Basic Info.:

 

Product Name: Tesamorelin

Unit Size: 2 mg/vial 

Unit Quantity: 1 Vial 

C6H9O-Tyr-Ala-Asp-Ala-Ile-Phe-Thr-Asn-Ser-Tyr-Arg-Lys-Val-Leu-Gly-Gln-Leu-Ser-Ala-Arg-Lys-Leu-Leu-Gln-Asp-Ile-Met-Ser-Arg-Gln-Gln-Gly-Glu-Ser-Asn-Gln-Glu-Arg-Gly-Ala-Arg-Ala-Arg-Leu-NH2

CAS: 218949-48-5

Molecular Formula: C211H366N72O67S1

Molecular Weight: 5135.89

Appearance: white powder

Purity (HPLC): ≥99.00%

Packing: According to every customer's requirement.

 

Tesamorelin Description:

 

Tesamorelin is a synthetic peptide consisting of all 44 amino acids of hGRF with the addition of a trans-3-Hexenoic acid group.Tesamorelin (also known as Egrifta) is a synthetic form of growth-hormone-releasing hormone which is used in the treatment of HIV-associated lipodystrophy.tendon fibroblasts in a dose-dependent manner as revealed by transwell filter migration assay. BPC 157 also dose dependently accelerated the spreading of tendon fibroblasts on culture dishes. The F-actin formation as detected by FITC-phalloidin staining was induced in BPC 157-treated fibroblasts. The protein expression and activation of FAK and paxillin were determined by Western blot analysis, and the phosphorylation levels of both FAK and paxillin were dose dependently increased by BPC 157 while the total amounts of protein was unaltered. In conclusion, BPC 157 promotes the ex vivo outgrowth of tendon fibroblasts from tendon explants, cell survival under stress, and the in vitro migration of tendon fibroblasts, which is likely mediated by the activation of the FAK-paxillin pathway.

 

Tesamorelin Applications:

 

1. Triptorelin raises testosterone levels by causing constant stimulation of the pituitary, it decreases pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle stimulating hormone (FSH). 

 

2. Like other GnRH agonists, triptorelin may be used in the treatment of hormone-responsive cancers such as prostate cancer or breast cancer, precocious puberty,estrogen-dependent conditions (such as endometriosis or uterine fibroids), and in assisted reproduction.