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High Purity Gw-501516 GW501516 For Weight Loss 317318-70-0

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High Purity Gw-501516 GW501516 For Weight Loss 317318-70-0
 
GW 501516 Basic Info:
 
Product Name: GW501516
Alias: Cardarine
CAS No.: 317318-70-0
Molecular Formula: C21H18F3NO3S2
Molecular Weight: 453.50
Purity: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Fat loss
Dose: The recommended dosage for GW is 10-20 mg and for 8 weeks length
 
GW 501516 Description:
 
GW501516 is the name of a Glaxo Wellcome drug (the GW stands for the company and the number
is that of the product). It is also known as GW-501,516, GW1516, GSK-516).
 
GW-501516 is a selective agonist with high affinity and it is very potent. Various studies on this
PPAR receptor in lab rats indicates that it regulates the various proteins that the body uses for
energy. Rats with high fat and low metabolism were given the product and they were able to
lose weight and to increase overall energy levels.
 
GW 501516 Application:
 
GW501516 (also known as GW-501,516, GW1516, GSK-516 and on the black market as Endurobol) is a PPARδ receptor agonist that was invented in a collaboration between Ligand Pharmaceuticals and GlaxoSmithKline in the 1990s, was entered into clinical development as a drug candidate for metabolic diseases and cardiovascular diseases, and was abandoned in 2007 because animal testing showed that the drug caused cancer to develop rapidly in several organs.
 
In 2007 research was published showing that high doses of GW501516 given to mice dramatically improved their physical performance; the work was widely discussed in popular media, and led to a black market for the drug candidate and to its abuse by athletes as a doping agent. The World Anti-Doping Agency (WADA) developed a test for GW501516 and other related chemicals and added them to the prohibited list in 2009; it has issued additional warnings to athletes that GW501516 is not safe.
 
History Of GW 501516:
 
Concerns were raised prior to the 2008 Beijing Olympics that GW501516 could be used by athletes as an ergogenic performance-enhancing drug that was not currently controlled by regulations or detected by standard tests. One of the main researchers from the study on enhanced endurance consequently developed a urine test to detect the drug, and made it available to the International Olympic Committee. The World Anti-Doping Agency (WADA) developed a test for GW501516 and other related PPARδ modulators,and added such drugs to the prohibited list in 2009.
 
GW501516 has been promoted on bodybuilding and athletics websites and by 2011 had already been available for some time on the black market. In 2011 it was reported to cost $1000 for 10 g.In 2012, WADA recategorised GW501516 from a gene doping compound to a "hormone and metabolic modulator".
 

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High Purity Male Hormone Raw Anabolic Trenbolone Steroids Mibolerone 3704-09-4

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High Purity Male Hormone Raw Anabolic Trenbolone Steroids Mibolerone 3704-09-4
 
Mibolerone Basic Info.:
 
Product Name: Mibolerone
CAS: 3704-09-4
MF: C20H30O2
MW: 302.45
EINECS: 223-046-5
Chemical Properties: White Crystalline Solid
Usage: Synthetic anabolic steroid related to testosterone. Controlled substance (anabolic steroid)
 
Mibolerone Description:
 
Mibolerone was initially as a veterinary product used to keep female dogs under control while they are in heat by shutting down the cycling of their ovaries. With proper timing, breeders are able to regulate the heat cycles of their bitches. Eventually, athletes began to utilize the product in order to boost aggression before events. It was even rumored that Mike Tyson was on Cheque Drops during the infamous ear biting incident during his bout with Holyfield. 
 
However, the late great guru Dan Duchaine discovered the application of Cheque Drops in modern bodybuilding far before that. The drops went in and out of production several times, before making a recent insurgence due to the piqued interest in the product thanks to the growing popularity of ultimate fighting circles.
 
Mibolerone Applications:
 
It is most commonly used by athletes about 30-40 minutes before their sporting event. Cheque drops are placed under the athletes tongue, and effects including aggression, strength and adrenaline rush are felt rapidly.  The drug leaves the body with in approximately four hours.
 
As well as being one of the most androgenic compounds, mibolerone is also one of the most toxic.   The most common side effect is progesterone related gynecomastia because it is a 19 nor-androgen.  
 

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High Purity Male Sex Hormones Sildenafil Mesylate For Male 131543-23-2

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High Purity Male Sex Hormones Sildenafil Mesylate For Male 131543-23-2
 
Sildenafil Mesylate Basic Info.:
 
Product Name: Sildenafil Mesylate
English name: Win 55,212-2 Mesylate
English Synonyms: Sildenafil Mesylate
CAS: 131543-23-2
MF: C28H30N2O6S
MW: 522.6126
Boiling point: 627.7 °C at 760 mmHg
Flash Point: 333.4 °C
Vapor Pressure: 1.14E-15mmHg at 25 °C
Properties:Solubility: 0.1 M HCl: 0.25 mg / mL
Appearance: White or white crystalline powder, odorless, bitter astringent taste, soluble in water and ethanol
Usage: Pharmaceutical raw materials, aphrodisiac It is medicine treatment raw material, indicated for the treatment of erectile dysfunction.
 
Sildenafil Mesylate Description:
 
Sildenafil Mesylate, same as Sildenafil is an inhibitor of type 5 -cGMP phosphodiesterase relaxing and smoothing muscle cells of the corpus cavernosum which leads to penile erection. This relaxation may be
mediated by nitric oxide via cyclic guanosine monophosphate.
 
pharmaceutical material, hormone. As a cyclic guanosine monophosphate (cGMP) specific phosphodiesterase type 5 (PDE5) selective inhibitor, penile smooth muscle relaxation allows rapid erection. Sildenafil is cheap, is the development and production of low-cost classes available kidney yang-like the perfect material for medicine and health products.
 
Sildenafil Mesylate Applications:
 
In 16 separate 4-24 week trials of men (over 18 years old) who suffered from impotence for longer than 6 months, dosages between 10-200 mgs were administered. Significant improvements in erectile function, including frequency of penetration as well as erection duration post penetration, were reported with Sildenfi* treatment compared to the placebo group.
Erections were improved in 72% of group verses 18% of the placebo group. In all cases effects were dependant upon dosage and improvement was the greatest when dosage exceeded 100 mgs. Responses were decreased by 40-60% in patients suffering from diabetes and prostatectomy, respectively. Withdrawal rates were less than 5% related to negative side effects and limited response rates
 

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High Purity Male Sex Hormones Vardenafil HCL / Levitra For Sex Enhancer Powder 224785-91-5

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High Purity Male Sex Hormones Vardenafil HCL / Levitra For Sex Enhancer Powder 224785-91-5
 
Vardenafil HCL Basic Info:
 
Product Name: 
Synonym: Fardenafil; Vardenafil hydrochloride
CAS No: 224785-91-5
MF: C23H33ClN6O4S
MW: 525.06
Purity: 99%
Melting point: 214-216°C
Half life: 4-5 hours
Appearance: White to Off-White Cyrstalline Solid, odorless, taste bitter and astringent soluble in water and alcohol.
Storage: in a cool and dry well-closed container and in ventilated area.
Product Categories: Intermediates & Fine Chemicals;Pharmaceuticals;Vardenafil
Usage: A selective phsphodiesterase type 5 (PDE5) inhibitor.
 
Vardenafil HCL Description:
 
Vardenafil (INN) is a PDE5 inhibitor used for treating erectile dysfunction. Vardenafil's indications and contra-indications are the same as with other PDE5 inhibitors; it is closely related in function to sildenafil citrate (Viagra) and tadalafil (Cialis). The difference between the vardenafil molecule and sildenafil citrate is a nitrogen atom's position and the change of sildenafil's piperazine ring methyl group to an ethyl group. Tadalafil is structurally different from both sildenafil and vardenafil. Vardenafil's relatively short effective time is comparable to but somewhat longer than sildenafil's.
 
Vardenafil HCL Application:
 
Beyond its indications for erectile dysfunction, vardenafil may be effective in the treatment of premature ejaculation, where it may significantly increase the time from vaginal penetration to ejaculation.Vardenafil, as with all PDE5 inhibitors, should not be used by men taking nitrate medications, because combining them with vardenafil might provoke potentially life-threatening hypotension (low blood pressure).
 
Further, Vardenafil causing lengthening of the QT interval. Therefore it should not be taken by men taking other medications that affect the QT interval (such as amiodarone).
 

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High Purity Natural API Heparin Sodium USP 93.3%min

Heparin Sodium is white or kind of white powder, odorless, has led to wet, soluble in water, insoluble in ethanol, acetone and other organic solvents.In aqueous solution, have a strong negative charge, can combine with some cation into molecular complex.A stable aqueous solution at pH 7., has the water absorbability.Anticoagulants physical and chemical properties of the molecular structure of heparin sodium heparin and low molecular heparin sodium drug interaction considerations heparin calcium heparin sodium reagent grade.


Formula: (C12H16NS2Na3) 20
Molecular weight: ca. 12000
EINECS No. : 232-681-7
Solubility: H2O: 50 mg/ml clear, faintly yellow
Form: crystalline (fine)
Color: white,
Merck: 14465 3
Stability: Stable. Incompatible with strong oxidizing agents, strong outside.
Than the curl: not less than 50 ° +
Ph: 5.5-8 .0
Protein: 0.5% or less
Dry weight loss: 5.0% or less
On ignition residue: 28.0 to 41.1%
Avoiding titer: 222 IU/mg
Wet product potency: 237 IU/mg
Packing: packed in aluminum drum
The physical and chemical properties: heparin sodium is white or kind of white powder, odorless, has led to wet, soluble in water, insoluble in ethanol, acetone and other organic solvents.in
In aqueous solution, have a strong negative charge, can combine with some cation into molecular complex.A stable aqueous solution at pH 7.

Heparin as anticoagulant drugs, it is a sticky polysaccharide substance, by extracted from the intestinal mucosa of pigs of glucosamine sulfate sodium salt, is secreted by the mast cells in human body and natural is present in the blood.Heparin sodium preventing platelet aggregation and destruction, inhibit fibrinogen to fibrin monomer, inhibit blood coagulation live element formation and confrontation of blood coagulation has been formed to live, blocking prothrombin into thrombin and antithrombin etc.
Heparin sodium in the body in vitro could delay or prevent blood clots.Its mechanism is very complex, on all affect the many steps in the process of blood coagulation.Its role as follows: (1) inhibit blood coagulation kinase of form and function, and thus hamper prothrombin into thrombin.(2) in relatively high concentrations of fashion has the inhibition of thrombin and other coagulation factors, the effect of preventing fibrinogen to fibrin;(3) can prevent platelet agglutination and destruction, etc.In addition, the anticoagulant effect of heparin sodium is its molecules associated with negative charge in the sulfuric acid root, has a positive charge, alkaline substances such as protamine or toluidine blue can neutralize the negative charges, so can inhibit its anticoagulant effect.Because of heparin in the body can activation and release of lipoprotein lipase, chyle particles of triglyceride and low density lipoprotein hydrolysis, so still have fall hematic fat action.
Heparin sodium can be used in the treatment of acute thromboembolic disease, diffuse intravascular coagulation (DIC).In recent years found that liver known as the removal of blood lipid.Deep intravenous or intramuscular injection or hypodermic, each unit of 5000 ~ 10000.Heparin of low toxicity, spontaneous bleeding tendency is the most main risk excessive use of heparin.Oral invalid and must be injected.Intramuscular injection or hypodermic stimulus is bigger, I can produce allergic reaction, even more than quantity can make cardiac arrest;I see a sex hair loss and diarrhea.In addition, the fair cause spontaneous fractures.Use for a long time sometimes can form thrombus, may be the consequences of anticoagulant enzyme - depletion.Has a tendency to bleeding, severe liver, renal insufficiency, severe hypertension, hemophilia, intracranial hemorrhage, peptic ulcer, pregnancy and postpartum, visceral tumors, trauma, and surgery are disabled heparin sodium.

 

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High Purity Nootropic Powder Fasoracetam 110958-19-5

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High Purity Nootropic Powder Fasoracetam 110958-19-5
 
Fasoracetam Basic Info.:
 
Product Name: Fasoracetam
Synonyms: Fasoracetam; Aka NS-105; LAM-105
CAS: 110958-19-5
MF: C10H16N2O2
MW: 196.248
EINECS: N/A
Product Categories: Pharmaceutical Intermediates; Nootropic Drug
 
Fasoracetam description:
 
Fasoracetam is a research compound and member of the racetam family of nootropics,primarily known for their cognitive enhancing abilities. Fasoracetam is also an anxiolytic and may be able to improve mood as well. This racetam works by affecting three receptors within the brain: acetylcholine,GABA and glutamate, all of three of which are involved in the creation and retention of memories.
 
it is now a nootropic smart drug which portrays itself in one of the most powerful racetams in the nootropic universe. Made from a class of compounds called the racetams, and acting on not only acetylcholine but also GABA receptors in the brain, this has the ability of activating both cholinergic and glutamate receptors of the cerebral cortex, and is a revolutionary racetam drug due to its extremely unique mechanism of action. Fasoracetam currently also shows benefits as an anti-depressant, ADHD stimulant, and an anxiolytic, it also, as proven in laboratories across the nation, helps with the formation and retention of new memories.
 
Fasoracetam has also been observed to block the amnestic effects of scopolamine in a rat model of cholinergic dysfunction, which was noted as an increase of both ACh release in the cerebral cortex, as well as HACU enhancement in both the cerebral cortex and hippocampus. ChAT activity remained unaffected. In the same study, Fasoracetam was able to reverse baclofen-induced memory disruption, thus suggesting a blocking role at the GABAB receptor.
 

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High Purity Nootropic Powder Picamilon / Pikamilone For Cognition Enhancer 34562-97-5

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High Purity Nootropic Powder Picamilon / Pikamilone For Cognition Enhancer 34562-97-5 
 
Pikamilone Basic Info.:
 
Product Name: Pikamilone
Synonyms: Pikamilone Hydrochloride;Nicotinoyl-Gaba;N-(3-Carboxypropyl) Nicotinamide;4-[(Pyridin-3-Ylcarbonyl)Amino]Butanoic Acid;4-(Nicotinamido)Butanoic Acid;Pikamiline;Pikamilone;
CAS: 34562-97-5
MF: C10H12N2O3
MW: 208.21
EINECS: N/A
Density: 1.245
Product Categories: Pharmaceutical Intermediates; Nootropic Drug; Heterocycles; Chemistry; API; Other APIs
Usage: anti-cancer agent; Used as a smart improve medicine
 
Picamilon Description:
What is the best way to use Picamilon powder and what Picamilon dosage should you be taking for optimal effects? This nootropic combination of GABA and Niacin offers a lot of cognitive benefits and mood enhancing effects. However, as an anxiolytic, it is often overlooked in favor of other nootropics like 
Sulbutiamine and Theanine. Picamilon is one of several Nootropic supplements that were originally developed in Russia (then called the Soviet Union) during the Cold War. This is probably why the supplement has been incredibly underused in the West for many years. Most of the studies and research were conducted and written in Russian, preventing its widespread dissemination even though Picamilon has been used since the early 1970′s. As such, it can be difficult to find usage and dosage information for this supplement online. In this article, we will tell you how to use Picamilon and what the recommended daily dose is. 
 
Picamilon Benefits:
The primary Nootropic benefits of this supplement center on mood boosting and overall brain function improvements. This includes helping to reduce feelings of stress and anxiety. In fact, many users feel that this supplement is so good at reducing these feelings that they use it on a regular basis to help relax. An improved positive outlook and attitude will also often follow. Once a person is relaxed, they will usually find themselves having improved sleep which is also more restful and deeper. As a brain booster, Picamilon benefits also include better mental energy and improved clarity and focus. It is easier to think and make decisions as well when using Picamilon supplements
 
Picamilon Function:
Picamilon is able to cross the blood-brain barrier and then is hydrolyzed into GABA and niacin. The released GABA in theory would activate GABA receptors potentially producing an anxiolytic response. The second released component, niacin acts as a strongvasodilator, which might be useful for the treatment of migraine headaches 
 
Picamilon Dosage:
The standard dosage range for Picamilon is between 50 and 300 mg per day.Of course, this may be split into several different administrations throughout the day, depending upon how it effects the user. Generally, a divided dose means one in the morning and one in the evening. Most supplements sell it in 150 mg tablets or capsules, but you can also buy it as a bulk powder to get more control over your dosages. Picamilon works best when taken on an empty stomach and the effects of this nootropic will last anywhere from two to four hours. You should always start out with the smallest effective Picamilon dose possible. Study the benefits obtained and then determine if increasing the dose is in order.
 
Stacking & Cycling Picamilon:
Many users have found that stacking and cycling their Picamilon dosages can be very effective. It is certainly very safe and it may even help to increase the effects of other Nootropic supplements like the Racetams including Aniracetam and Piracetam. There are a number of other Nootropics that have similar effects to Picamilon, but might lead to tolerance if used on a daily basis. This means that it might be helpful to include Picamilon as part of a cycle with something like, say, 
Start with the safer option (Picamilon) and use on a 3 or 4 day on and 2 day off cycle. For the days off of Picamilon, substitute with the 
 

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High Purity Nootropics Powder Adrafinils 63547-13-7

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High Purity Nootropics Powder Adrafinils 63547-13-7

Adrafinil Basic information

Product Name: Adrafinil

Synonyms: 2-((diphenylmethyl)sulfinyl)-acetohydroxamicaci;2-((diphenylmethyl)sulfinyl)-n-hydroxy-acetamid;2-((diphenylmethyl)sulfinyl)-n-hydroxyacetamide;2-(benzhydrylsulfinyl)acetohydroxamicacid;ADRAFINIL;2-[(DIPHENYLMETHYL)SULFINYL]ACETOHYDROXAMIC ACID;CRL 40028;OLMIFON

CAS: 63547-13-7

MF: C15H15NO3S

MW: 289.35

EINECS: 264-303-1

Melting point: 159-1600C

Storage temp.: -20°C Freezer

Solubility: DMSO: 35 mg/mL

Chemical Properties: Light Pink Solid

Usage: a-Adrenergic agonist. Treatment of depression

Product Categories: Aromatics Compounds;Aromatics;Intermediates & Fine Chemicals;Pharmaceuticals;Sulfur & Selenium Compounds.

 

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High Purity Pharmaceutical Intermediates Dehydroepiandrosterone Acetate 853-23-6

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High Purity Pharmaceutical Intermediates Dehydroepiandrosterone Acetate 853-23-6
 
Dehydroepiandrosterone Acetate Basic Info.:
 
Product Name: Dehydroepiandrosterone Acetate
Synonyms: Dehydroepiandrosterone Acetate;Dehydroepiandrosterone-3-Acetate;Dehydroisoandrosterone 3-Acetate;Dehydroisoandrosterone Acetate;Dehydroisoandrosterone Acetate;Prasterone Acetate
CAS: 853-23-6
MF: C21H30O3
MW: 330.46
EINECS: 212-714-1
Purity: 99%
Melting point: 168-170 °C(lit.)
Storage temp.: Refrigerator
Chemical Properties: Off-White Solid
Usage: Menopausal syndrome;A metabolite of Dehydroepiandrosterone. This mammalian pro-hormone promotes brain and immune function
Product Categories: Pharmaceutical Intermediates;Steroids;17-Ketosteroids;Biochemistry;Hydroxyketosteroids;Chemistry;Intermediates & Fine Chemicals;Metabolites & Impurities;Pharmaceuticals;API;Inhibitors
 

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High Purity Pharmaceutical Raw Materials UDCA Powder Ursodeoxycholic Acid 128-13-2

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High Purity Pharmaceutical Raw Materials UDCA Powder Ursodeoxycholic Acid 128-13-2
 
Ursodeoxycholic Acid Basic Info.:
 
Product Name: Ursodeoxycholic Acid
EINECS: 204-879-3
CAS Registry Number: 128-13-2
Molecular Formula: C24H40O4
Molecular Weight: 392.58
Appearance: White crystalline powder
Application: For the prevention treatment of choles.
PackAge: Foil bag or drum
Production Capacity: 5000 Kilogram/Month
Purity: 99%
Storage: Sealed, light and oxygen resistant
 
Ursodeoxycholic Acid Description:
 
Ursodeoxycholic Acid is white powder,almost insoluble in water,freely soluble in alcohol.
Ursodeoxycholic acid (UDCA), also known as ursodiol, is a compound produced from bile by the action of intestinal bacteria. Since this bile acid is not produced directly by the body, it is known as a secondary bile acid.One of the functions of bile acids is to act in the intestine to help digest fats and fatsoluble vitamins from food.
Ursodeoxycholic acid has been used in pharmacology to dissolve gallstones made of cholesterol, and to treat liver disorders. It has been used for a long time in both human and veterinary medicine.
 
Ursodeoxycholic Acid Application:
 
UDCA Powder Ursodeoxycholic Acid Can increase the secretion of bile acid.
UDCA Powder Ursodeoxycholic Acid Reduce cholesterol in bile and cholesterol ester.
UDCA Powder Ursodeoxycholic Acid Is conducive to the cholesterol gradually dissolve gallstones.
UDCA Powder Ursodeoxycholic Acid Should not be used for surgical treatment of cholesterol stone, but cannot dissolve the bile pigment stone, mixing and opaque X line of stones.
 

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